If you made any changes in Pure these will be visible here soon.

Fingerprint Dive into the research topics where Eiji Kawanishi is active. These topic labels come from the works of this person. Together they form a unique fingerprint.

Network Recent external collaboration on country level. Dive into details by clicking on the dots.

Research Output

  • 542 Citations
  • 12 h-Index
  • 19 Article
  • 1 Review article

Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety

Koizumi, Y., Tanaka, Y., Matsumura, T., Kadoh, Y., Miyoshi, H., Hongu, M., Takedomi, K., Kotera, J., Sasaki, T., Taniguchi, H., Watanabe, Y., Takakuwa, M., Kojima, K., Baba, N., Nakamura, I. & Kawanishi, E., Aug 1 2019, In : Bioorganic and Medicinal Chemistry. 27, 15, p. 3440-3450 11 p.

Research output: Contribution to journalArticle

  • 2 Citations (Scopus)

    Scalable Process Design for a PDE10A Inhibitor Consisting of Pyrazolopyrimidine and Quinoxaline as Key Units

    Yamagami, T., Kobayashi, R., Moriyama, N., Horiuchi, H., Toyofuku, E., Kadoh, Y., Kawanishi, E., Izumoto, S., Hiramatsu, H., Nanjo, T., Sugino, M., Utsugi, M. & Moritani, Y., Apr 19 2019, In : Organic Process Research and Development. 23, 4, p. 578-587 10 p.

    Research output: Contribution to journalArticle

  • 2 Citations (Scopus)

    Discovery of 2-[(E)-2-(7-fluoro-3-methylquinoxalin-2-yl)vinyl]-6-pyrrolidin- 1-yl-N-(tetrahydro-2H-pyran-4-yl)pyrimidin-4-amine hydrochloride as a highly selective PDE10A inhibitor

    Kadoh, Y., Miyoshi, H., Matsumura, T., Tanaka, Y., Hongu, M., Kimura, M., Takedomi, K., Omori, K., Kotera, J., Sasaki, T., Kobayashi, T., Taniguchi, H., Watanabe, Y., Kojima, K., Sakamoto, T., Himiyama, T. & Kawanishi, E., 2018, In : Chemical and Pharmaceutical Bulletin. 66, 3, p. 243-250 8 p.

    Research output: Contribution to journalArticle

  • 4 Citations (Scopus)

    Synthetic Method for 2′-Amino-LNA Bearing Any of the Four Nucleobases via a Transglycosylation Reaction

    Sawamoto, H., Arai, Y., Yamakoshi, S., Obika, S. & Kawanishi, E., Apr 6 2018, In : Organic Letters. 20, 7, p. 1928-1931 4 p.

    Research output: Contribution to journalArticle

  • 2 Citations (Scopus)

    Computation-assisted disconnection approach for the synthesis of neoantimycins, 15-membered macrocyclic depsipeptides

    Yamakoshi, S., Okamoto, M., Sawamoto, H., Arai, Y., Kawanishi, E., Sasaki, M. & Takeda, K., Mar 1 2017, In : Current Organic Synthesis. 14, 2, p. 299-308 10 p.

    Research output: Contribution to journalArticle

  • 2 Citations (Scopus)