Abstract
The title compound was produced diastereoselectively in racemic and optically active forms by employing the [2 + 2] cycloaddition reaction of an imine with benzyloxyketene followed by acidic alcoholysis of the formed 3,4-cis-disubstituted β-lactam with isopropanol.
| Original language | English |
|---|---|
| Pages (from-to) | 299-302 |
| Number of pages | 4 |
| Journal | Heterocycles |
| Volume | 30 |
| Issue number | 1 |
| Publication status | Published - Jan 1 1990 |
| Externally published | Yes |
Fingerprint
All Science Journal Classification (ASJC) codes
- Analytical Chemistry
- Pharmacology
- Organic Chemistry
Cite this
A novel synthesis of cyclohexylnorstatine isopropyl ester, the C-terminal component of a renin inhibitor. / Ito, Yoshio; Kamijo, Tetsuhide; Harada, Hiromu; Terashima, Shiro.
In: Heterocycles, Vol. 30, No. 1, 01.01.1990, p. 299-302.Research output: Contribution to journal › Article
}
TY - JOUR
T1 - A novel synthesis of cyclohexylnorstatine isopropyl ester, the C-terminal component of a renin inhibitor
AU - Ito, Yoshio
AU - Kamijo, Tetsuhide
AU - Harada, Hiromu
AU - Terashima, Shiro
PY - 1990/1/1
Y1 - 1990/1/1
N2 - The title compound was produced diastereoselectively in racemic and optically active forms by employing the [2 + 2] cycloaddition reaction of an imine with benzyloxyketene followed by acidic alcoholysis of the formed 3,4-cis-disubstituted β-lactam with isopropanol.
AB - The title compound was produced diastereoselectively in racemic and optically active forms by employing the [2 + 2] cycloaddition reaction of an imine with benzyloxyketene followed by acidic alcoholysis of the formed 3,4-cis-disubstituted β-lactam with isopropanol.
UR - http://www.scopus.com/inward/record.url?scp=0142199048&partnerID=8YFLogxK
UR - http://www.scopus.com/inward/citedby.url?scp=0142199048&partnerID=8YFLogxK
M3 - Article
AN - SCOPUS:0142199048
VL - 30
SP - 299
EP - 302
JO - Heterocycles
JF - Heterocycles
SN - 0385-5414
IS - 1
ER -