A practical one-pot synthesis of 2,3-disubstituted indoles from unactivated anilines

Makoto Tokunaga; Mitsuru Ota; Masa aki Haga; Yasuo Wakatsuki

doi:10.1016/S0040-4039(01)00588-3

A practical one-pot synthesis of 2,3-disubstituted indoles from unactivated anilines

Makoto Tokunaga, Mitsuru Ota, Masa aki Haga, Yasuo Wakatsuki

Research output: Contribution to journal › Article › peer-review

65 Citations (Scopus)

Abstract

2-Substituted-3-methyl indoles are synthesized with good regioselectivity from readily available substrates and catalysts, i.e. the reaction of anilines with propargyl alcohols in the presence of 0.36-1 mol% Ru₃(CO)₁₂.

Original language	English
Pages (from-to)	3865-3868
Number of pages	4
Journal	Tetrahedron Letters
Volume	42
Issue number	23
DOIs	https://doi.org/10.1016/S0040-4039(01)00588-3
Publication status	Published - Jun 4 2001
Externally published	Yes

All Science Journal Classification (ASJC) codes

Biochemistry
Drug Discovery
Organic Chemistry

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10.1016/S0040-4039(01)00588-3

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title = "A practical one-pot synthesis of 2,3-disubstituted indoles from unactivated anilines",

abstract = "2-Substituted-3-methyl indoles are synthesized with good regioselectivity from readily available substrates and catalysts, i.e. the reaction of anilines with propargyl alcohols in the presence of 0.36-1 mol% Ru3(CO)12.",

author = "Makoto Tokunaga and Mitsuru Ota and Haga, {Masa aki} and Yasuo Wakatsuki",

year = "2001",

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doi = "10.1016/S0040-4039(01)00588-3",

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T1 - A practical one-pot synthesis of 2,3-disubstituted indoles from unactivated anilines

AU - Tokunaga, Makoto

AU - Ota, Mitsuru

AU - Haga, Masa aki

AU - Wakatsuki, Yasuo

PY - 2001/6/4

Y1 - 2001/6/4

N2 - 2-Substituted-3-methyl indoles are synthesized with good regioselectivity from readily available substrates and catalysts, i.e. the reaction of anilines with propargyl alcohols in the presence of 0.36-1 mol% Ru3(CO)12.

AB - 2-Substituted-3-methyl indoles are synthesized with good regioselectivity from readily available substrates and catalysts, i.e. the reaction of anilines with propargyl alcohols in the presence of 0.36-1 mol% Ru3(CO)12.

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DO - 10.1016/S0040-4039(01)00588-3

M3 - Article

AN - SCOPUS:0035806306

SN - 0040-4039

VL - 42

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JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 23

ER -

A practical one-pot synthesis of 2,3-disubstituted indoles from unactivated anilines

Abstract

All Science Journal Classification (ASJC) codes

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