Abstract
The meta-selective introduction of functional groups into aromatic substrates was successfully achieved by hydrogen-bond-controlled meta-selective C-H borylation and successive conversion of the boryl group to other functional groups. By this method a wide range of functional groups could be introduced without isolation of the borylated intermediates. The desired meta-functionalized aromatic products were obtained in a one-pot manner even on a gram scale. Regioselective synthesis of multisubstituted aromatic compounds was also achieved.
Original language | English |
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Pages (from-to) | 1342-1346 |
Number of pages | 5 |
Journal | Organic letters |
Volume | 21 |
Issue number | 5 |
DOIs | |
Publication status | Published - Mar 1 2019 |
All Science Journal Classification (ASJC) codes
- Biochemistry
- Physical and Theoretical Chemistry
- Organic Chemistry