Oxetanyl peptides: Novel peptidomimetic modules for medicinal chemistry

Martin McLaughlin, Ryo Yazaki, Thomas C. Fessard, Erick M. Carreira

Research output: Contribution to journalArticlepeer-review

41 Citations (Scopus)


The synthesis of novel oxetanyl peptides, where the amide bond is replaced by a non-hydrolyzable oxetanylamine fragment, is reported. This new class of pseudo-dipeptides with the same H-bond donor/acceptor pattern found in proteins expands the repertoire of peptidomimetics.

Original languageEnglish
Pages (from-to)4070-4073
Number of pages4
JournalOrganic letters
Issue number16
Publication statusPublished - Aug 15 2014
Externally publishedYes

All Science Journal Classification (ASJC) codes

  • Biochemistry
  • Physical and Theoretical Chemistry
  • Organic Chemistry


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