Tuned Classical Thermal Aromatization Furnishing an Estrogenic Benzoacridine

Rintaro Koga, Tohru Oishi, Kohei Torikai

Research output: Contribution to journalArticle

1 Citation (Scopus)

Abstract

The diversity-oriented doubling strategy, which generates two 12-arylbenzoacridines from a single triarylmethanol precursor was developed to construct a library of drug candidates for the identification of biologically active compounds. Exploration of this 12-arylbenzoacridine library furnished a 4′-OH derivative as an estrogenic compound.

Original languageEnglish
Article numberst-2015-s0585-c
Pages (from-to)2801-2805
Number of pages5
JournalSynlett
Volume26
Issue number20
DOIs
Publication statusPublished - Dec 17 2015

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Aromatization
Estrogens
Derivatives
Pharmaceutical Preparations
Hot Temperature

All Science Journal Classification (ASJC) codes

  • Organic Chemistry

Cite this

Tuned Classical Thermal Aromatization Furnishing an Estrogenic Benzoacridine. / Koga, Rintaro; Oishi, Tohru; Torikai, Kohei.

In: Synlett, Vol. 26, No. 20, st-2015-s0585-c, 17.12.2015, p. 2801-2805.

Research output: Contribution to journalArticle

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