Boronic Acid Accelerated Three-Component Reaction for the Synthesis of α-Sulfanyl-Substituted Indole-3-acetic Acids

Amrita Das, Kenji Watanabe, Hiroyuki Morimoto, Takashi Ohshima

研究成果: ジャーナルへの寄稿記事

10 引用 (Scopus)

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Boronic acid was used to accelerate a three-component reaction of indoles, thiols, and glyoxylic acids for the synthesis of α-sulfanyl-substituted indole-3-acetic acids. Boronic acid catalysis to activate the α-hydroxy group in α-hydroxycarboxylic acid intermediates and intramolecular assistance by free carboxylic acid were the keys to accelerating the product formation.

元の言語英語
ページ(範囲)5794-5797
ページ数4
ジャーナルOrganic Letters
19
発行部数21
DOI
出版物ステータス出版済み - 11 3 2017

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All Science Journal Classification (ASJC) codes

  • Biochemistry
  • Physical and Theoretical Chemistry
  • Organic Chemistry

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