Synthesis and Insecticidal Activity of Oxazaphospholidines, Oxathiaphospholanes, and Thiazaphospholidines

Wu Shao-Yong, Akinori Hirashima, Ryuko Takeya, Morifusa Eto

研究成果: ジャーナルへの寄稿記事

2 引用 (Scopus)

抄録

Fifty-five new five-membered cyclic organophosphorus compounds including oxazaphospholidines, thiazaphospholidines, and oxathiaphospholanes were synthesized, which have substituents at 4- or/and 5-positions besides at the 2-position. The thiazaphospholidines showed the highest insecticidal activity followed by oxathiaphospholanes and oxazaphospholidines. The position preference of substituents in insecticidal activity was most obvious in the oxazaphospholidines. It was preferable for insecticidal activity to have the substituent near the more basic atom: the 4-position for thiazaphospholidine and oxazaphospholidine, the 5-position for oxathiaphospholane, with the exception of 4- or 5-phenyl oxazaphospholidine.

元の言語英語
ページ(範囲)2911-2917
ページ数7
ジャーナルAgricultural and Biological Chemistry
52
発行部数11
DOI
出版物ステータス出版済み - 1 1 1988

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organophosphorus compounds
synthesis
Organophosphorus Compounds
Atoms
oxathiaphospholane

All Science Journal Classification (ASJC) codes

  • Biochemistry, Genetics and Molecular Biology(all)
  • Agricultural and Biological Sciences(all)

これを引用

Synthesis and Insecticidal Activity of Oxazaphospholidines, Oxathiaphospholanes, and Thiazaphospholidines. / Shao-Yong, Wu; Hirashima, Akinori; Takeya, Ryuko; Eto, Morifusa.

:: Agricultural and Biological Chemistry, 巻 52, 番号 11, 01.01.1988, p. 2911-2917.

研究成果: ジャーナルへの寄稿記事

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